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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Oxidized low-density lipoprotein receptor 1
(Bovine)
Pharmaxis
US Patent
Ligand
BDBM454323
((Z)-2-(1-(4-amino-2-fluorobut-2-en-1-yl- 2-methyl-...)
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Affinity Data
IC50: >300nM
Assay Description:
LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Lysyl oxidase homolog 2
(Homo sapiens (Human))
Pharmaxis
US Patent
Ligand
BDBM454323
((Z)-2-(1-(4-amino-2-fluorobut-2-en-1-yl- 2-methyl-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: <300nM
Assay Description:
LOX: The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the i...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Oxidized low-density lipoprotein receptor 1
(Bovine)
Pharmaxis
US Patent
Ligand
BDBM454323
((Z)-2-(1-(4-amino-2-fluorobut-2-en-1-yl- 2-methyl-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >300nM
Assay Description:
LOX: The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the i...
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Lysyl oxidase homolog 2
(Homo sapiens (Human))
Pharmaxis
US Patent
Ligand
BDBM454323
((Z)-2-(1-(4-amino-2-fluorobut-2-en-1-yl- 2-methyl-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: <300nM
Assay Description:
LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI