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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146474(CHEMBL419896 | N-{2-(1,4-Dioxa-spiro[4.5]dec-8-yl)...)
Affinity DataIC50:  60nMAssay Description:Inhibition of Tumor necrosis factor alpha converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-17(Homo sapiens (Human))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146474(CHEMBL419896 | N-{2-(1,4-Dioxa-spiro[4.5]dec-8-yl)...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of matrix metalloproteinase-17More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146474(CHEMBL419896 | N-{2-(1,4-Dioxa-spiro[4.5]dec-8-yl)...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146474(CHEMBL419896 | N-{2-(1,4-Dioxa-spiro[4.5]dec-8-yl)...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of matrix metalloproteinase-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146474(CHEMBL419896 | N-{2-(1,4-Dioxa-spiro[4.5]dec-8-yl)...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of matrix metalloproteinase-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Kaken Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50146474(CHEMBL419896 | N-{2-(1,4-Dioxa-spiro[4.5]dec-8-yl)...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of matrix metalloproteinase-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed