Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetALK tyrosine kinase receptor(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50294549(1-Chloro-3-methyl-5-phenethyl-5,6,7,12-tetrahydro-...)
Affinity DataIC50:  1.18E+4nMAssay Description:Inhibition of 6xHis-tagged human NPM-ALK expressed in insect cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50294549(1-Chloro-3-methyl-5-phenethyl-5,6,7,12-tetrahydro-...)
Affinity DataIC50:  1.24E+4nMAssay Description:Inhibition of recombinant METMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50294549(1-Chloro-3-methyl-5-phenethyl-5,6,7,12-tetrahydro-...)
Affinity DataIC50:  1.26E+4nMAssay Description:Inhibition of recombinant IGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50294549(1-Chloro-3-methyl-5-phenethyl-5,6,7,12-tetrahydro-...)
Affinity DataIC50:  1.98E+4nMAssay Description:Inhibition of human recombinant IRKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
St. Jude Children'S Research Hospital

Curated by ChEMBL
LigandPNGBDBM50294549(1-Chloro-3-methyl-5-phenethyl-5,6,7,12-tetrahydro-...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of recombinant JAK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed