Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 12 hits in this display
BDBM421843(7-(2-(4-(4-(1-Methyl-1H-1,2,4-triazol-3-yl)phenyl)...)
BDBM421843(7-(2-(4-(4-(1-Methyl-1H-1,2,4-triazol-3-yl)phenyl)...)
IC50: <50nMAssay Description:Activated ERK1 and ERK2 activity was determined in a Mobility Shift Assay (MSA) format as follows: Compound and kinase solution were prepared with as...More data for this Ligand-Target Pair
BDBM421845((S)-7-(2-(4-(4-(1-Methyl-1H-1,2,4-triazol-3-yl)phe...)IC50: <50nMAssay Description:Activated ERK1 and ERK2 activity was determined in a Mobility Shift Assay (MSA) format as follows: Compound and kinase solution were prepared with as...More data for this Ligand-Target Pair
BDBM421845((S)-7-(2-(4-(4-(1-Methyl-1H-1,2,4-triazol-3-yl)phe...)
IC50: <50nMAssay Description:Activated ERK1 and ERK2 activity was determined in a Mobility Shift Assay (MSA) format as follows: Compound and kinase solution were prepared with as...More data for this Ligand-Target Pair
BDBM421846((R)-7-(2-(4-(4-(1-Methyl-1H-1,2,4-triazol-3-yl)phe...)IC50: <50nMAssay Description:Activated ERK1 and ERK2 activity was determined in a Mobility Shift Assay (MSA) format as follows: Compound and kinase solution were prepared with as...More data for this Ligand-Target Pair
BDBM421845((S)-7-(2-(4-(4-(1-Methyl-1H-1,2,4-triazol-3-yl)phe...)
BDBM421846((R)-7-(2-(4-(4-(1-Methyl-1H-1,2,4-triazol-3-yl)phe...)
IC50: <50nMAssay Description:Activated ERK1 and ERK2 activity was determined in a Mobility Shift Assay (MSA) format as follows: Compound and kinase solution were prepared with as...More data for this Ligand-Target Pair
BDBM421843(7-(2-(4-(4-(1-Methyl-1H-1,2,4-triazol-3-yl)phenyl)...)
IC50: <50nMAssay Description:Activated ERK1 and ERK2 activity was determined in a Mobility Shift Assay (MSA) format as follows: Compound and kinase solution were prepared with as...More data for this Ligand-Target Pair
BDBM421843(7-(2-(4-(4-(1-Methyl-1H-1,2,4-triazol-3-yl)phenyl)...)
IC50: <50nMAssay Description:Activated ERK1 and ERK2 activity was determined in a Mobility Shift Assay (MSA) format as follows: Compound and kinase solution were prepared with as...More data for this Ligand-Target Pair
BDBM421845((S)-7-(2-(4-(4-(1-Methyl-1H-1,2,4-triazol-3-yl)phe...)
IC50: <50nMAssay Description:Activated ERK1 and ERK2 activity was determined in a Mobility Shift Assay (MSA) format as follows: Compound and kinase solution were prepared with as...More data for this Ligand-Target Pair
BDBM421846((R)-7-(2-(4-(4-(1-Methyl-1H-1,2,4-triazol-3-yl)phe...)
IC50: 150nMAssay Description:Activated ERK1 and ERK2 activity was determined in a Mobility Shift Assay (MSA) format as follows: Compound and kinase solution were prepared with as...More data for this Ligand-Target Pair
BDBM421846((R)-7-(2-(4-(4-(1-Methyl-1H-1,2,4-triazol-3-yl)phe...)
IC50: 150nMAssay Description:Activated ERK1 and ERK2 activity was determined in a Mobility Shift Assay (MSA) format as follows: Compound and kinase solution were prepared with as...More data for this Ligand-Target Pair