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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University Of Tennessee Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50412062(CHEMBL294755)
Affinity DataKi:  15.1nMAssay Description:Inhibition of human ENT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Toxoplasma gondii)TBA
LigandPNGBDBM50412062(CHEMBL294755)
Affinity DataKi:  3.30E+3nMAssay Description:Inhibition of Toxoplasma gondii adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University Of Tennessee Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50412062(CHEMBL294755)
Affinity DataIC50:  457nMAssay Description:Binding affinity to ENT1 transporterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Toxoplasma gondii)TBA
LigandPNGBDBM50412062(CHEMBL294755)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of Toxoplasma gondii adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAdenosine kinase(Toxoplasma gondii)TBA
LigandPNGBDBM50412062(CHEMBL294755)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of Toxoplasma gondii adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article