Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 16 hits in this display
BDBM107698(US11426393, Compound Table XV.4 | US8598210, Table...)
BDBM107698(US11426393, Compound Table XV.4 | US8598210, Table...)
BDBM107698(US11426393, Compound Table XV.4 | US8598210, Table...)
BDBM107698(US11426393, Compound Table XV.4 | US8598210, Table...)
BDBM107698(US11426393, Compound Table XV.4 | US8598210, Table...)
BDBM107698(US11426393, Compound Table XV.4 | US8598210, Table...)
IC50: 650nMAssay Description:Inhibition of recombinant human PHD2 (179 to 426 residues) using HIF-1alpha (556 to 574 residues) as substrate after 20 mins by MALDI-TOF MS analysisMore data for this Ligand-Target Pair
BDBM107698(US11426393, Compound Table XV.4 | US8598210, Table...)
IC50: 650nMAssay Description:The EGLN-1 (or EGLN-3) enzyme activity is determined using mass spectrometry (matrix-assisted laser desorption ionization, time-of-flight MS, MALDI-T...More data for this Ligand-Target Pair
BDBM107698(US11426393, Compound Table XV.4 | US8598210, Table...)
IC50: 650nMT: 2°CAssay Description:The EGLN-1 (or EGLN-3) enzyme activity is determined using mass spectrometry (matrix-assisted laser desorption ionization, time-of-flight MS, MALDI-T...More data for this Ligand-Target Pair
BDBM107698(US11426393, Compound Table XV.4 | US8598210, Table...)
IC50: 650nMAssay Description:The EGLN-1 (or EGLN-3) enzyme activity is determined using mass spectrometry (matrix-assisted laser desorption ionization, time-of-flight MS, MALDI-T...More data for this Ligand-Target Pair
BDBM107698(US11426393, Compound Table XV.4 | US8598210, Table...)
IC50: 650nMAssay Description:The EGLN-1 (or EGLN-3) enzyme activity is determined using mass spectrometry (matrix-assisted laser desorption ionization, time-of-flight MS, MALDI-T...More data for this Ligand-Target Pair
BDBM107698(US11426393, Compound Table XV.4 | US8598210, Table...)
BDBM107698(US11426393, Compound Table XV.4 | US8598210, Table...)
BDBM107698(US11426393, Compound Table XV.4 | US8598210, Table...)
BDBM107698(US11426393, Compound Table XV.4 | US8598210, Table...)
BDBM107698(US11426393, Compound Table XV.4 | US8598210, Table...)
BDBM107698(US11426393, Compound Table XV.4 | US8598210, Table...)