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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetHuntingtin(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM54857(3-[4-[(Z)-3-(4-bromophenyl)-3-keto-prop-1-enyl]-3-...)
Affinity DataIC50:  2.60E+3nMMore data for this Ligand-Target Pair
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TargetM17 leucyl aminopeptidase(Plasmodium falciparum 3D7)
Srmlsc

Curated by PubChem BioAssay
LigandPNGBDBM54857(3-[4-[(Z)-3-(4-bromophenyl)-3-keto-prop-1-enyl]-3-...)
Affinity DataIC50:  3.40E+4nMAssay Description:Southern Research Molecular Libraries Screening Center (SRMLSC) Southern Research Institute (Birmingham, Alabama) NIH Molecular Libraries Screening...More data for this Ligand-Target Pair
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TargetStreptokinase A(Streptococcus pyogenes M1 GAS)
Broad Institute

Curated by PubChem BioAssay
LigandPNGBDBM54857(3-[4-[(Z)-3-(4-bromophenyl)-3-keto-prop-1-enyl]-3-...)
Affinity DataEC50:  3.53E+3nMAssay Description:Keywords: Group A streptococcus, GAS, streptokinase, expression, virulence, inhibition, dose response, EC50 Assay Overview: The goal of this assa...More data for this Ligand-Target Pair
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TargetSerine/threonine-protein kinase 33(Homo sapiens (Human))
Broad Institute

Curated by PubChem BioAssay
LigandPNGBDBM54857(3-[4-[(Z)-3-(4-bromophenyl)-3-keto-prop-1-enyl]-3-...)
Affinity DataEC50:  1.93E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
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TargetStreptokinase A(Streptococcus pyogenes M1 GAS)
Broad Institute

Curated by PubChem BioAssay
LigandPNGBDBM54857(3-[4-[(Z)-3-(4-bromophenyl)-3-keto-prop-1-enyl]-3-...)
Affinity DataEC50:  2.33E+3nMAssay Description:Keywords: Group A streptococcus, GAS, streptokinase, expression, virulence, inhibition, dose response, EC50 Assay Overview: The goal of this assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay