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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Gamma-aminobutyric acid receptor subunit alpha-1
(Rattus norvegicus (Rat))
Lund University
Curated by
ChEMBL
Ligand
BDBM50293264
(2-(5-bromo-2-hydroxyphenyl)-6-methylquinolin-4(1H)...)
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Affinity Data
Ki: 39nM
Assay Description:
Displacement of [3H]flumazenil in rat GABAAalpha1beta3gamma2 receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Gamma-aminobutyric acid receptor subunit alpha-3
(RAT)
Lund University
Curated by
ChEMBL
Ligand
BDBM50293264
(2-(5-bromo-2-hydroxyphenyl)-6-methylquinolin-4(1H)...)
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Copy InChI
Affinity Data
Ki: 99nM
Assay Description:
Displacement of [3H]flumazenil in rat GABAAalpha3beta3gamma2 receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Gamma-aminobutyric acid receptor subunit alpha-2
(Rattus norvegicus (Rat))
Lund University
Curated by
ChEMBL
Ligand
BDBM50293264
(2-(5-bromo-2-hydroxyphenyl)-6-methylquinolin-4(1H)...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 120nM
Assay Description:
Displacement of [3H]flumazenil in rat GABAAalpha2beta3gamma2 receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI