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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
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Target
Equilibrative nucleoside transporter 2
(Homo sapiens (Human))
Monash University Malaysia
Curated by
ChEMBL
Ligand
BDBM56941
(6-[[4-(4-fluorophenyl)-1-piperazinyl]methyl]-N2-(3...)
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Affinity Data
IC50: 570nM
Assay Description:
Inhibition of human ENT2 transfected in nucleoside transporter-deficient pig PK-15 cells assessed as inhibition of [3H]-uridine uptake by liquid scin...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
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PubMed
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Target
Equilibrative nucleoside transporter 1
(Homo sapiens (Human))
Monash University Malaysia
Curated by
ChEMBL
Ligand
BDBM56941
(6-[[4-(4-fluorophenyl)-1-piperazinyl]methyl]-N2-(3...)
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Affinity Data
IC50: 2.38E+3nM
Assay Description:
Inhibition of human ENT1 transfected in nucleoside transporter-deficient pig PK-15 cells assessed as inhibition of [3H]-uridine uptake by liquid scin...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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PubMed
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Target
Streptokinase A
(Streptococcus pyogenes M1 GAS)
Broad Institute
Curated by
PubChem BioAssay
Ligand
BDBM56941
(6-[[4-(4-fluorophenyl)-1-piperazinyl]methyl]-N2-(3...)
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Affinity Data
EC50: 1.50E+5nM
Assay Description:
Keywords: Group A streptococcus, GAS, streptokinase, expression, virulence, inhibition, dose response, EC50 Assay Overview: The goal of this assa...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Similars
In Depth
Details
PCBioAssay
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