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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetEquilibrative nucleoside transporter 2(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM56941(6-[[4-(4-fluorophenyl)-1-piperazinyl]methyl]-N2-(3...)
Affinity DataIC50:  570nMAssay Description:Inhibition of human ENT2 transfected in nucleoside transporter-deficient pig PK-15 cells assessed as inhibition of [3H]-uridine uptake by liquid scin...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM56941(6-[[4-(4-fluorophenyl)-1-piperazinyl]methyl]-N2-(3...)
Affinity DataIC50:  2.38E+3nMAssay Description:Inhibition of human ENT1 transfected in nucleoside transporter-deficient pig PK-15 cells assessed as inhibition of [3H]-uridine uptake by liquid scin...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetStreptokinase A(Streptococcus pyogenes M1 GAS)
Broad Institute

Curated by PubChem BioAssay
LigandPNGBDBM56941(6-[[4-(4-fluorophenyl)-1-piperazinyl]methyl]-N2-(3...)
Affinity DataEC50:  1.50E+5nMAssay Description:Keywords: Group A streptococcus, GAS, streptokinase, expression, virulence, inhibition, dose response, EC50 Assay Overview: The goal of this assa...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay