Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 7 hits in this display
BDBM26791(benzimidazole analog., 17 | tert-butyl (3S,4S)-3-(...)
BDBM26791(benzimidazole analog., 17 | tert-butyl (3S,4S)-3-(...)
Ki: 2.61E+3nM ΔG°: -31.9kJ/molepH: 7.5 T: 2°CAssay Description:The compounds were tested for enzyme inhibition using fluorescence resonance energy transfer (FRET) assay. Fluorescence measurements were performed i...More data for this Ligand-Target Pair
BDBM26791(benzimidazole analog., 17 | tert-butyl (3S,4S)-3-(...)
Matrilysin(Homo sapiens (Human))Bristol-Myers Squibb
BDBM26791(benzimidazole analog., 17 | tert-butyl (3S,4S)-3-(...)
Ki: 5.86E+3nM ΔG°: -29.9kJ/molepH: 7.5 T: 2°CAssay Description:The compounds were tested for enzyme inhibition using fluorescence resonance energy transfer (FRET) assay. Fluorescence measurements were performed i...More data for this Ligand-Target Pair
BDBM26791(benzimidazole analog., 17 | tert-butyl (3S,4S)-3-(...)
IC50: 1nMpH: 7.5 T: 2°CAssay Description:The compounds were tested for enzyme inhibition using fluorescence resonance energy transfer (FRET) assay. Fluorescence measurements were performed i...More data for this Ligand-Target Pair
BDBM26791(benzimidazole analog., 17 | tert-butyl (3S,4S)-3-(...)
IC50: 250nMpH: 7.5 T: 2°CAssay Description:The compounds were tested for enzyme inhibition using fluorescence resonance energy transfer (FRET) assay. Fluorescence measurements were performed i...More data for this Ligand-Target Pair
BDBM26791(benzimidazole analog., 17 | tert-butyl (3S,4S)-3-(...)
IC50: 1.60E+3nMAssay Description:The compounds were tested for enzyme inhibition using fluorescence resonance energy transfer (FRET) assay. Fluorescence measurements were performed i...More data for this Ligand-Target Pair