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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
8
hits in this display
Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM50116515
(CHEMBL3609729)
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Affinity Data
EC50: 4nM
Assay Description:
Positive allosteric modulator activity at human mGlu4 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
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CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
PDB
3D Structure (crystal)
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Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM50116515
(CHEMBL3609729)
Copy SMILES
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Affinity Data
EC50: 9nM
Assay Description:
Positive allosteric modulator activity at rat mGlu4 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
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CHEMBL
PC cid
PC sid
PDB
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In Depth
Details
Article
PubMed
PDB
3D Structure (crystal)
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Target
Metabotropic glutamate receptor 7
(Rattus norvegicus (Rat))
Vanderbilt University
Curated by
ChEMBL
Ligand
BDBM50116515
(CHEMBL3609729)
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Affinity Data
EC50: >1.00E+4nM
Assay Description:
Positive allosteric modulation of rat mGlu7 receptor expressed in HEK cells co-expressing Galphai5 assessed as increase in glutamate-induced calcium ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Metabotropic glutamate receptor 8
(Homo sapiens (Human))
TBA
Ligand
BDBM50116515
(CHEMBL3609729)
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Affinity Data
EC50: 1.20E+3nM
Assay Description:
Positive allosteric modulation of mGluR8 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
PubMed
Copy BDB DOI
Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM50116515
(CHEMBL3609729)
Copy SMILES
Copy InChI
Affinity Data
EC50: 52nM
Assay Description:
Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells co-expressing Gqi5 assessed as increase in glutamate-induced calcium mo...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
PDB
3D Structure (crystal)
Copy BDB DOI
Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Massachusetts General Hospital
Curated by
ChEMBL
Ligand
BDBM50116515
(CHEMBL3609729)
Copy SMILES
Copy InChI
Affinity Data
EC50: 52nM
Assay Description:
Positive allosteric modulation of mGluR4 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
PubMed
PDB
3D Structure (crystal)
Copy BDB DOI
Target
Metabotropic glutamate receptor 7
(Homo sapiens (Human))
TBA
Ligand
BDBM50116515
(CHEMBL3609729)
Copy SMILES
Copy InChI
Affinity Data
EC50: >1.00E+4nM
Assay Description:
Positive allosteric modulation of mGluR7 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
PubMed
Copy BDB DOI
Target
Metabotropic glutamate receptor 8
(Rattus norvegicus (Rat))
Vanderbilt University
Curated by
ChEMBL
Ligand
BDBM50116515
(CHEMBL3609729)
Copy SMILES
Copy InChI
Affinity Data
EC50: 1.20E+3nM
Assay Description:
Positive allosteric modulation of rat mGlu8 receptor expressed in HEK cells co-expressing Galphai5 assessed as increase in glutamate-induced calcium ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI