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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440162(CHEMBL2426591)
Affinity DataIC50:  92nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Mus musculus)
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440162(CHEMBL2426591)
Affinity DataIC50:  255nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed