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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136419(3,4-Dichloro-N-(2-oxo-1,2,3,4-tetrahydro-quinolin-...)
Affinity DataIC50:  1.37E+3nMAssay Description:Inhibitory concentration against recombinant human liver glycogen phosphorylase a (HLGPa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136419(3,4-Dichloro-N-(2-oxo-1,2,3,4-tetrahydro-quinolin-...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50136419(3,4-Dichloro-N-(2-oxo-1,2,3,4-tetrahydro-quinolin-...)
Affinity DataIC50:  2.31E+3nMAssay Description:Inhibitory concentration against recombinant human muscle glycogen phosphorylase a (HMGPa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed