Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 11 hits in this display   

TargetDual specificity protein kinase CLK4(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50259404(CHEMBL4076448)
Affinity DataIC50:  190nMAssay Description:Inhibition of GST tagged recombinant mouse CLK4 expressed in Escherichia coli using RS peptide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50259404(CHEMBL4076448)
Affinity DataIC50:  310nMAssay Description:Inhibition of GST tagged recombinant mouse CLK1 expressed in Escherichia coli using RS peptide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50259404(CHEMBL4076448)
Affinity DataIC50:  650nMAssay Description:Inhibition of GST tagged recombinant human DYRK1A expressed in Escherichia coli using woodtide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50259404(CHEMBL4076448)
Affinity DataIC50:  820nMAssay Description:Inhibition of human recombinant CDK5/p25 after 30 mins by [gamma-33P]ATP based scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50259404(CHEMBL4076448)
Affinity DataIC50:  820nMAssay Description:Inhibition of GST tagged recombinant human DYRK2 expressed in Escherichia coli using using woodtide as substrate after 30 mins by [gamma-33P]ATP base...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50259404(CHEMBL4076448)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of GST tagged recombinant mouse CLK2 expressed in Escherichia coli using RS peptide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50259404(CHEMBL4076448)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of GST tagged recombinant human DYRK3 expressed in Escherichia coli using woodtide as substrate after 30 mins by [gamma-33P]ATP based scin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50259404(CHEMBL4076448)
Affinity DataIC50:  2.10E+3nMAssay Description:In vitro inhibition of [3H]DAMGO binding to Opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50259404(CHEMBL4076448)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of human recombinant CDK9/cyclin T expressed in insect cells using CDK7/9-tide as substrate after 30 mins by [gamma-33P]ATP based scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK3(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50259404(CHEMBL4076448)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GST tagged recombinant mouse CLK3 expressed in Escherichia coli using RS peptide as substrate after 30 mins by [gamma-33P]ATP based sci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50259404(CHEMBL4076448)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 after 30 mins by [gamma-33P]ATP based scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed