Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL

LigandBDBM50289535(CHEMBL4176184)Copy SMILESCopy InChI

Affinity DataEC50:  7.90E+3nMAssay Description:Potentiator activity at CFTR F508-del mutant (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPurchaseChEBI
PC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of Genoa

Curated by ChEMBL

LigandBDBM50289535(CHEMBL4176184)Copy SMILESCopy InChI

Affinity DataEC50:  1.60E+4nMAssay Description:Corrector activity at CFTR F508-del mutant (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPurchaseChEBI
PC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI