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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50432003(CHEMBL2348740)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant CDK5/p25 after 30 mins by scintillation counting analysis in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50432003(CHEMBL2348740)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat recombinant DYRK1A expressed in Escherichia coli using myelin basic protein as substrate after 30 mins by scintillation counting an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Sus scrofa)
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50432003(CHEMBL2348740)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of pig brain CK1 using RRKHAAIGpSAYSITA as substrate after 30 mins by scintillation counting analysis in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed