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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Cystic fibrosis transmembrane conductance regulator
(Homo sapiens (Human))
University Of California
Curated by
ChEMBL
Ligand
BDBM50353339
(CHEMBL1831059)
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Affinity Data
IC50: 100nM
Assay Description:
Inhibition of human wild-type CFTR expressed in FRT cells assessed as inhibition of forskolin-induced short-circuit current by voltage clamp electrop...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Cystic fibrosis transmembrane conductance regulator
(Homo sapiens (Human))
University Of California
Curated by
ChEMBL
Ligand
BDBM50353339
(CHEMBL1831059)
Copy SMILES
Copy InChI
Affinity Data
IC50: 170nM
Assay Description:
Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI