Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Decode Chemistry

Curated by ChEMBL
LigandPNGBDBM50247939(3-(4-(3,4-dichlorophenoxy)-1-methyl-1H-indol-3-yl)...)
Affinity DataIC50:  12.4nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor at 20 uM in presence of normal bufferMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Decode Chemistry

Curated by ChEMBL
LigandPNGBDBM50247939(3-(4-(3,4-dichlorophenoxy)-1-methyl-1H-indol-3-yl)...)
Affinity DataIC50:  50.8nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor at 20 uM in presence of 10% human serumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Decode Chemistry

Curated by ChEMBL
LigandPNGBDBM50247939(3-(4-(3,4-dichlorophenoxy)-1-methyl-1H-indol-3-yl)...)
Affinity DataIC50:  2.40E+3nMAssay Description:Displacement of radioligand from FP receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Decode Chemistry

Curated by ChEMBL
LigandPNGBDBM50247939(3-(4-(3,4-dichlorophenoxy)-1-methyl-1H-indol-3-yl)...)
Affinity DataIC50:  4.20E+3nMAssay Description:Displacement of radioligand from EP2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Decode Chemistry

Curated by ChEMBL
LigandPNGBDBM50247939(3-(4-(3,4-dichlorophenoxy)-1-methyl-1H-indol-3-yl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of radioligand from EP1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Decode Chemistry

Curated by ChEMBL
LigandPNGBDBM50247939(3-(4-(3,4-dichlorophenoxy)-1-methyl-1H-indol-3-yl)...)
Affinity DataIC50:  2.04E+4nMAssay Description:Displacement of radioligand from EP4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed