Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 8 hits in this display
BDBM247367(US9447092, Comparator 1, Example 56)
BDBM247367(US9447092, Comparator 1, Example 56)
IC50: 30nMAssay Description:Inhibition of CYP isozymes was determined using a mixture of probe substrates. The samples were incubated for 10 minutes followed by protein precipit...More data for this Ligand-Target Pair
BDBM247367(US9447092, Comparator 1, Example 56)
IC50: 30nMAssay Description:Inhibition of CYP isozymes was determined using a mixture of probe substrates. The samples were incubated for 10 minutes followed by protein precipit...More data for this Ligand-Target Pair
BDBM247367(US9447092, Comparator 1, Example 56)
BDBM247367(US9447092, Comparator 1, Example 56)
IC50: <1.00E+3nMAssay Description:Inhibition of CYP isozymes was determined using a mixture of probe substrates. The samples were incubated for 10 minutes followed by protein precipit...More data for this Ligand-Target Pair
BDBM247367(US9447092, Comparator 1, Example 56)
BDBM247367(US9447092, Comparator 1, Example 56)
IC50: 3.00E+4nMAssay Description:Inhibition of CYP isozymes was determined using a mixture of probe substrates. The samples were incubated for 10 minutes followed by protein precipit...More data for this Ligand-Target Pair
BDBM247367(US9447092, Comparator 1, Example 56)
IC50: >5.00E+4nMAssay Description:Inhibition of CYP isozymes was determined using a mixture of probe substrates. The samples were incubated for 10 minutes followed by protein precipit...More data for this Ligand-Target Pair