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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Celgene Quantscel Research

US Patent
LigandPNGBDBM381941(2-{1-methyl-5-[4- (trifluoromethoxy)phenyl]-1H- im...)
Affinity DataIC50:  550nMAssay Description:The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 2B(Homo sapiens (Human))
Celgene Quantscel Research

US Patent
LigandPNGBDBM381941(2-{1-methyl-5-[4- (trifluoromethoxy)phenyl]-1H- im...)
Affinity DataIC50:  550nMAssay Description:The ability of test compounds to inhibit the activity of FBXL10 was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Celgene Quantscel Research

US Patent
LigandPNGBDBM381941(2-{1-methyl-5-[4- (trifluoromethoxy)phenyl]-1H- im...)
Affinity DataIC50:  550nMAssay Description:The ability of test compounds to inhibit the activity of Jarid1B was determined in 384-well plate format under the following reaction conditions: 0.8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
Celgene Quantscel Research

US Patent
LigandPNGBDBM381941(2-{1-methyl-5-[4- (trifluoromethoxy)phenyl]-1H- im...)
Affinity DataIC50:  5.50E+3nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent