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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
EF-hand calcium-binding domain-containing protein 4B
(Homo sapiens (Human))
Rhizen Pharmaceuticals
US Patent
Ligand
BDBM141409
(US10668051, Compound Example 49 | US8921364, 49)
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Affinity Data
IC50: 65.5nM
T: 2°C
Assay Description:
Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat # T9033) induced endoplasmic calcium release in Jurkat cells. (see Yasu...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
US Patent
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Target
Calcium release-activated calcium channel protein 1
(Homo sapiens (Human))
Rhizen Pharmaceuticals
US Patent
Ligand
BDBM141409
(US10668051, Compound Example 49 | US8921364, 49)
Copy SMILES
Copy InChI
Affinity Data
IC50: 65.5nM
Assay Description:
Inhibition of CRAC channels was determined following thapsigargin (Sigma, Cat #T9033) induced endoplasmic calcium release in Jurkat cells, (see Yasur...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI