Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 8 hits in this display
BDBM361347(6-((1H-pyrazolo[4,3-b] pyridin- 3-yl)amino)-N-(3,3...)
BDBM361347(6-((1H-pyrazolo[4,3-b] pyridin- 3-yl)amino)-N-(3,3...)
BDBM361347(6-((1H-pyrazolo[4,3-b] pyridin- 3-yl)amino)-N-(3,3...)
BDBM361347(6-((1H-pyrazolo[4,3-b] pyridin- 3-yl)amino)-N-(3,3...)
BDBM361347(6-((1H-pyrazolo[4,3-b] pyridin- 3-yl)amino)-N-(3,3...)
BDBM361347(6-((1H-pyrazolo[4,3-b] pyridin- 3-yl)amino)-N-(3,3...)
EC50: 50nMAssay Description:Positive allosteric modulation of human mGlu4 receptor expressed in CHO cells co-expressing Gqi5 assessed as increase in glutamate-induced calcium mo...More data for this Ligand-Target Pair
BDBM361347(6-((1H-pyrazolo[4,3-b] pyridin- 3-yl)amino)-N-(3,3...)
BDBM361347(6-((1H-pyrazolo[4,3-b] pyridin- 3-yl)amino)-N-(3,3...)