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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM50247868(2-(3-Chloro-4-fluorophenyl)isothiazol-3(2H)-one | ...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of human recombinant HAT PCAFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Horizon Discovery

Curated by ChEMBL
LigandPNGBDBM50247868(2-(3-Chloro-4-fluorophenyl)isothiazol-3(2H)-one | ...)
Affinity DataIC50:  6.10E+3nMAssay Description:Binding affinity to GST-tagged Pin1 (unknown origin) by SPR spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed