Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
D3-Pharmachemistry

Curated by ChEMBL
LigandPNGBDBM50561341(CHEMBL4745672)
Affinity DataEC50:  96nMAssay Description:Potentiation of human CFTR F508 deletion mutant expressed in rat FRT cells coexpressing HS-YFP assessed as increase in iodide influx pre-incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed