Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 15 hits in this display
BDBM397147(US10596172, Compound I-28 | US10828300, Compound I...)
BDBM397147(US10596172, Compound I-28 | US10828300, Compound I...)
BDBM397147(US10596172, Compound I-28 | US10828300, Compound I...)
IC50: <10nMAssay Description:Briefly, 10× stocks of EGFR-WT (PV3872) from Invitrogen and EGFR-T790M/L858R (40350) from BPS Bioscience, San Diego, Calif., 1.13×ATP (AS001A) and ap...More data for this Ligand-Target Pair
BDBM397147(US10596172, Compound I-28 | US10828300, Compound I...)
BDBM397147(US10596172, Compound I-28 | US10828300, Compound I...)
IC50: <10nMAssay Description:Briefly, 10× stocks of EGFR-WT (PV3872) from Invitrogen and EGFR-T790M/L858R (40350) from BPS Bioscience, San Diego, Calif., 1.13×ATP (AS001A) and ap...More data for this Ligand-Target Pair
BDBM397147(US10596172, Compound I-28 | US10828300, Compound I...)
BDBM397147(US10596172, Compound I-28 | US10828300, Compound I...)
IC50: 55nMAssay Description:Briefly, 10× stocks of EGFR-WT (PV3872) from Invitrogen and EGFR-T790M/L858R (40350) from BPS Bioscience, San Diego, Calif., 1.13×ATP (AS001A) and ap...More data for this Ligand-Target Pair
BDBM397147(US10596172, Compound I-28 | US10828300, Compound I...)
IC50: 55nMAssay Description:Briefly, 10× stocks of EGFR-WT (PV3872) from Invitrogen and EGFR-T790M/L858R (40350) from BPS Bioscience, San Diego, Calif., 1.13×ATP (AS001A) and ap...More data for this Ligand-Target Pair
BDBM397147(US10596172, Compound I-28 | US10828300, Compound I...)
BDBM397147(US10596172, Compound I-28 | US10828300, Compound I...)
BDBM397147(US10596172, Compound I-28 | US10828300, Compound I...)
BDBM397147(US10596172, Compound I-28 | US10828300, Compound I...)
IC50: <100nMAssay Description:Briefly, 10x stocks of EGFR-WT (PV3872) from Invitrogen and EGFR-T790M/L858R (40350) from BPS Bioscience, San Diego, Calif., 1.13×ATP (AS001A) and ap...More data for this Ligand-Target Pair
BDBM397147(US10596172, Compound I-28 | US10828300, Compound I...)
IC50: <100nMAssay Description:Briefly, 10x stocks of EGFR-WT (PV3872) from Invitrogen and EGFR-T790M/L858R (40350) from BPS Bioscience, San Diego, Calif., 1.13×ATP (AS001A) and ap...More data for this Ligand-Target Pair
BDBM397147(US10596172, Compound I-28 | US10828300, Compound I...)
IC50: 550nMAssay Description:Briefly, 10x stocks of EGFR-WT (PV3872) from Invitrogen and EGFR-T790M/L858R (40350) from BPS Bioscience, San Diego, Calif., 1.13×ATP (AS001A) and ap...More data for this Ligand-Target Pair
BDBM397147(US10596172, Compound I-28 | US10828300, Compound I...)
IC50: 550nMAssay Description:Briefly, 10x stocks of EGFR-WT (PV3872) from Invitrogen and EGFR-T790M/L858R (40350) from BPS Bioscience, San Diego, Calif., 1.13×ATP (AS001A) and ap...More data for this Ligand-Target Pair