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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM50089516
((1R,2S)-1-amino-2-(phosphonomethyl)cyclopropanecar...)
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Affinity Data
EC50: 580nM
Assay Description:
Agonistic activity at Metabotropic glutamate receptor 4 expressed in mammalian cells by GTPgammaS binding assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Metabotropic glutamate receptor 8
(Homo sapiens (Human))
University Paris Descartes
Curated by
ChEMBL
Ligand
BDBM50089516
((1R,2S)-1-amino-2-(phosphonomethyl)cyclopropanecar...)
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Affinity Data
EC50: 6.51E+3nM
Assay Description:
Agonist activity at mGlu8 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate production
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Metabotropic glutamate receptor 7
(Homo sapiens (Human))
University Paris Descartes
Curated by
ChEMBL
Ligand
BDBM50089516
((1R,2S)-1-amino-2-(phosphonomethyl)cyclopropanecar...)
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Affinity Data
EC50: >3.00E+6nM
Assay Description:
Agonist activity at mGlu7 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate production
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM50089516
((1R,2S)-1-amino-2-(phosphonomethyl)cyclopropanecar...)
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Copy InChI
Affinity Data
EC50: 4.08E+4nM
Assay Description:
Agonist activity at mGlu4 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate production
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Metabotropic glutamate receptor 6
(Homo sapiens (Human))
University Paris Descartes
Curated by
ChEMBL
Ligand
BDBM50089516
((1R,2S)-1-amino-2-(phosphonomethyl)cyclopropanecar...)
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Affinity Data
EC50: 1.11E+5nM
Assay Description:
Agonist activity at mGlu6 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate production
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI