Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetLarge neutral amino acids transporter small subunit 1(Homo sapiens (Human))
University Of Nebraska At Kearney

Curated by ChEMBL

LigandBDBM50463209(CHEMBL4249170)Copy SMILESCopy InChI

Affinity DataIC50:  1.00E+5nMAssay Description:Cis-inhibition of human LAT1 expressed in TREx HEK293 cells assessed as inhibition of [3H]-gabapentin uptake preincubated for 3 mins at 37 degC follo...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPurchasePC cidPC sidPDB

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetLarge neutral amino acids transporter small subunit 1(Homo sapiens (Human))
University Of Nebraska At Kearney

Curated by ChEMBL

LigandBDBM50463209(CHEMBL4249170)Copy SMILESCopy InChI

Affinity DataIC50:  1.00E+5nMAssay Description:Cis-inhibition of human LAT1 expressed in TREx HEK293 cells at 200 uM assessed as inhibition of [3H]-gabapentin uptake preincubated for 3 mins at 37 ...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPurchasePC cidPC sidPDB

In DepthDetails ArticlePubMed
Copy BDB DOI