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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50109655(2-Amino-3-(3-hydroxy-4-naphthalen-1-yl-isoxazol-5-...)
Affinity DataKi:  6.20E+4nMAssay Description:The compound was tested for the receptor binding affinity at Metabotropic glutamate receptor 5 using established second messenger assay systems.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50109655(2-Amino-3-(3-hydroxy-4-naphthalen-1-yl-isoxazol-5-...)
Affinity DataKi:  1.19E+5nMAssay Description:The compound was tested for the receptor binding affinity at Metabotropic glutamate receptor 1 using established second messenger assay systems.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50109655(2-Amino-3-(3-hydroxy-4-naphthalen-1-yl-isoxazol-5-...)
Affinity DataKi: >1.00E+6nMAssay Description:The compound was tested for the receptor binding affinity at Metabotropic glutamate receptor 4 using established second messenger assay systems.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50109655(2-Amino-3-(3-hydroxy-4-naphthalen-1-yl-isoxazol-5-...)
Affinity DataKi: >1.00E+6nMAssay Description:The compound was tested for the receptor binding affinity at Metabotropic glutamate receptor 2 using established second messenger assay systems.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
The Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50109655(2-Amino-3-(3-hydroxy-4-naphthalen-1-yl-isoxazol-5-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration of the compound which causes 50% reduction in receptor binding affinity against Ionotropic glutamate receptor ionotropic kainate using ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed