Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetCollagenase 3(Homo sapiens (Human))
Graz University Of Technology

Curated by ChEMBL

LigandBDBM50607144(CHEMBL5219839)Copy SMILESCopy InChI

Affinity DataIC50:  18nMAssay Description:Inhibition of recombinant human MMP13 using APMA and fTHP-15(FAM) as substrate preincubated for 30 mins followed by substrate addition by fluorescenc...More data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails PubMed
Copy BDB DOI

Target72 kDa type IV collagenase(Homo sapiens (Human))
Graz University Of Technology

Curated by ChEMBL

LigandBDBM50607144(CHEMBL5219839)Copy SMILESCopy InChI

Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of MMP-2 (unknown origin) using fTHP-15(FAM) as substrateMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails PubMed
Copy BDB DOI