Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetProtein kinase C theta type(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL

LigandBDBM50573012(CHEMBL4878146)Copy SMILESCopy InChI

Affinity DataIC50:  150nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetProtein kinase C delta type(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL

LigandBDBM50573012(CHEMBL4878146)Copy SMILESCopy InChI

Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of PKA-delta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI