Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetArginase-1(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50316605(2-amino-5-(2-aminoimidazol-4-yl)pentanoic acid | C...)
Affinity DataKi: >8.00E+7nMAssay Description:Inhibition of human recombinant full length arginase 1 expressed in Escherichia coli BL21(DE3) by fixed point assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50316605(2-amino-5-(2-aminoimidazol-4-yl)pentanoic acid | C...)
Affinity DataIC50:  6.50E+4nMAssay Description:Inhibition of mouse recombinant iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Rattus norvegicus (rat))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50316605(2-amino-5-(2-aminoimidazol-4-yl)pentanoic acid | C...)
Affinity DataIC50:  6.50E+4nMAssay Description:Inhibition rat recombinant nNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed