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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetGlycogen phosphorylase, muscle form(Homo sapiens (Human))
University Of Alcala

Curated by ChEMBL
LigandPNGBDBM50077949(2-Aminomethyl-6-hydroxymethyl-tetrahydro-pyran-3,4...)
Affinity DataKi:  1.78E+6nMAssay Description:Inhibitory activity against rabbit muscle glycogen phosphorylaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Homo sapiens (Human))
University Of Alcala

Curated by ChEMBL
LigandPNGBDBM50077949(2-Aminomethyl-6-hydroxymethyl-tetrahydro-pyran-3,4...)
Affinity DataKi:  1.78E+6nMAssay Description:Inhibitory activity against rabbit muscle glycogen phosphorylaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
Philipps-Universit£T Marburg

Curated by ChEMBL
LigandPNGBDBM50473933(CHEMBL1161038)
Affinity DataKi:  1.58E+7nMAssay Description:Inhibitory activity against Pig Skeletal Glycogen Phosphorylase bMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
Philipps-Universit£T Marburg

Curated by ChEMBL
LigandPNGBDBM50077949(2-Aminomethyl-6-hydroxymethyl-tetrahydro-pyran-3,4...)
Affinity DataKi:  1.68E+7nMAssay Description:Inhibition of rabbit glycogen phosphorylase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
Philipps-Universit£T Marburg

Curated by ChEMBL
LigandPNGBDBM50077949(2-Aminomethyl-6-hydroxymethyl-tetrahydro-pyran-3,4...)
Affinity DataKi:  1.68E+7nMAssay Description:Inhibition of rabbit glycogen phosphorylase B enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
Philipps-Universit£T Marburg

Curated by ChEMBL
LigandPNGBDBM50147894((S)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-py...)
Affinity DataKi:  1.68E+7nMAssay Description:Inhibitory binding constant against glycogen phosphorylase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
Philipps-Universit£T Marburg

Curated by ChEMBL
LigandPNGBDBM50473931(CHEMBL1161041)
Affinity DataKi:  3.16E+7nMAssay Description:Inhibitory activity against Pig Skeletal Glycogen Phosphorylase bMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, brain form(Homo sapiens (Human))
Philipps-Universit£T Marburg

Curated by ChEMBL
LigandPNGBDBM50147884((R)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-py...)
Affinity DataKi:  3.45E+7nMAssay Description:Inhibitory binding constant against glycogen phosphorylase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed