Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 34 hits in this display
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
IC50: >1.00E+3nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
IC50: >1.00E+3nMAssay Description:LOX: The assay was developed using either 384 or 96 well format. Briefly, in a standard 384 well plate assay 25 μL of a dilution of any of the i...More data for this Ligand-Target Pair
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
BDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)
IC50: <1.00E+6nMAssay Description:LOX and LOXL2: Lysyl oxidase (LOX) is an extracellular copper dependent enzyme which oxidizes peptidyl lysine and hydroxylysine residues in collagen ...More data for this Ligand-Target Pair