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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287143(6-Amino-2-{2-benzyl-3-[((R)-1-benzyloxycarbonylami...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of endothelin-converting enzyme in human umbilical vein endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287143(6-Amino-2-{2-benzyl-3-[((R)-1-benzyloxycarbonylami...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of endothelin-converting enzyme in human umbilical vein endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287143(6-Amino-2-{2-benzyl-3-[((R)-1-benzyloxycarbonylami...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of neutral endopeptidase in human umbilical vein endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287143(6-Amino-2-{2-benzyl-3-[((R)-1-benzyloxycarbonylami...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of neutral endopeptidase in human umbilical vein endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails Article