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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
MAP kinase-interacting serine/threonine-protein kinase 1
(Homo sapiens (Human))
A*Star
Curated by
ChEMBL
Ligand
BDBM152261
(US8993552, 4H8 Compound 42)
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Affinity Data
IC50: 1.40E+4nM
Assay Description:
Inhibition of N-terminal GST-tagged MNK1 (unknown origin) (37 to 341 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
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PDB
In Depth
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Article
PubMed
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Target
MAP kinase-interacting serine/threonine-protein kinase 2
(Homo sapiens (Human))
A*Star
Curated by
ChEMBL
Ligand
BDBM152261
(US8993552, 4H8 Compound 42)
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Affinity Data
IC50: 1.70E+4nM
Assay Description:
Inhibition of N-terminal GST-tagged MNK2 (unknown origin) (72 to 385 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
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PC cid
PC sid
PDB
In Depth
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Article
PubMed
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Target
Menin
(Homo sapiens (Human))
University of Michigan
US Patent
Ligand
BDBM152261
(US8993552, 4H8 Compound 42)
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Affinity Data
IC50: 5.00E+4nM
Assay Description:
Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
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PDB
In Depth
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US Patent
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Target
Tyrosine-protein kinase receptor UFO
(Homo sapiens (Human))
Experimental Drug Development Centre
Curated by
ChEMBL
Ligand
BDBM152261
(US8993552, 4H8 Compound 42)
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Affinity Data
IC50: 3.63E+5nM
Assay Description:
Inhibition of Axl (unknown origin) using 5'FAM labeled KKKKEEIYFFF-NH2 peptide as substrate incubated for 1.5 hrs
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
PDB
In Depth
Details
Article
PubMed
Copy BDB DOI