Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetCasein kinase I isoform delta(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50563723(CHEMBL4128865)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of wild-type human CK1delta using PLSRTLpSVASLPGL as substrate incubated for 40 mins in presence of ATP by Kinase-Glo luminescence assayMore data for this Ligand-Target Pair
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50563723(CHEMBL4128865)
Affinity DataIC50:  17nMAssay Description:Inhibition of wild-type human CK1epsilon using PLSRTLpSVASLPGL as substrate incubated for 70 mins in presence of ATP by Kinase-Glo luminescence assayMore data for this Ligand-Target Pair