Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 7 hits in this display
BDBM50049823(4-Amino-7-((2R,3R,4S,5R)-3,4-dihydroxy-5-hydroxyme...)
BDBM50049823(4-Amino-7-((2R,3R,4S,5R)-3,4-dihydroxy-5-hydroxyme...)
BDBM50049823(4-Amino-7-((2R,3R,4S,5R)-3,4-dihydroxy-5-hydroxyme...)
BDBM50049823(4-Amino-7-((2R,3R,4S,5R)-3,4-dihydroxy-5-hydroxyme...)
IC50: 4.40E+4nMAssay Description:Inhibition of DOT1L (unknown origin) using chicken nucleosome as substrate in presence of [3H]SAM incubated for 1 hr by TopCount methodMore data for this Ligand-Target Pair
BDBM50049823(4-Amino-7-((2R,3R,4S,5R)-3,4-dihydroxy-5-hydroxyme...)
BDBM50049823(4-Amino-7-((2R,3R,4S,5R)-3,4-dihydroxy-5-hydroxyme...)
BDBM50049823(4-Amino-7-((2R,3R,4S,5R)-3,4-dihydroxy-5-hydroxyme...)