Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 5 hits in this display
Caspase-6(Homo sapiens (Human))Washington University
BDBM29572(isatin Michael acceptor (IMA) analogue, 11a)
Caspase-3(Homo sapiens (Human))Washington University
BDBM29572(isatin Michael acceptor (IMA) analogue, 11a)
Caspase-7(Homo sapiens (Human))Washington University
BDBM29572(isatin Michael acceptor (IMA) analogue, 11a)
Caspase-1(Homo sapiens (Human))Washington University
BDBM29572(isatin Michael acceptor (IMA) analogue, 11a)
Caspase-8(Homo sapiens (Human))Washington University
BDBM29572(isatin Michael acceptor (IMA) analogue, 11a)
IC50: >5.00E+4nMpH: 7.4 T: 2°CAssay Description:The caspase enzymatic activity was determined by measuring the accumulation of a fluorogenic product. All assays were prepared in 96-well format. Rec...More data for this Ligand-Target Pair