Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetHistone deacetylase 3(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50089658(CHEMBL3577299)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant HDAC3 using MAZ1600 as fluorogenic substrate measured every 5 mins by optimized homogenous fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50089658(CHEMBL3577299)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant HDAC2 using MAZ1600 as fluorogenic substrate measured every 5 mins by optimized homogenous fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50089658(CHEMBL3577299)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant HDAC8 using MAZ1675 as fluorogenic substrate measured every 5 mins by optimized homogenous fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50089658(CHEMBL3577299)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant HDAC6 using MAZ1600 as fluorogenic substrate measured every 5 mins by optimized homogenous fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50089658(CHEMBL3577299)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant HDAC1 using MAZ1600 as fluorogenic substrate measured every 5 mins by optimized homogenous fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed