Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 4 hits in this display
BDBM154602(US8999957, Column 162-163, Compound 1 | US8999957,...)
BDBM154602(US8999957, Column 162-163, Compound 1 | US8999957,...)
IC50: 591nMAssay Description:Condition 1: Activated ERK2 activity was also determined in the IMAP assay format using the procedure outlined above. 1 μl of 25× compound was a...More data for this Ligand-Target Pair
BDBM154602(US8999957, Column 162-163, Compound 1 | US8999957,...)
BDBM154602(US8999957, Column 162-163, Compound 1 | US8999957,...)
Kd: 9.20nMAssay Description:The SAR (Structure Activity Relationship) for ERK ligands covered by this invention was interrogated using the TdF (Temperature Dependence Fluorescen...More data for this Ligand-Target Pair