Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 4 hits in this display
Kallikrein-7(Homo sapiens (Human))Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Ki: 1.80E+3nMAssay Description:Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Ki: 7.07E+4nMAssay Description:Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Kallikrein-7(Homo sapiens (Human))Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
IC50: 1.33E+4nMAssay Description:Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
IC50: 9.92E+4nMAssay Description:Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair