Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 20 hits in this display
BDBM24776(1,4-Naphthoquinone | 1,4-Naphthoquinone (5a) | 1,4...)
BDBM24776(1,4-Naphthoquinone | 1,4-Naphthoquinone (5a) | 1,4...)
BDBM24776(1,4-Naphthoquinone | 1,4-Naphthoquinone (5a) | 1,4...)
BDBM24776(1,4-Naphthoquinone | 1,4-Naphthoquinone (5a) | 1,4...)
BDBM24776(1,4-Naphthoquinone | 1,4-Naphthoquinone (5a) | 1,4...)
BDBM24776(1,4-Naphthoquinone | 1,4-Naphthoquinone (5a) | 1,4...)
BDBM24776(1,4-Naphthoquinone | 1,4-Naphthoquinone (5a) | 1,4...)
BDBM24776(1,4-Naphthoquinone | 1,4-Naphthoquinone (5a) | 1,4...)
BDBM24776(1,4-Naphthoquinone | 1,4-Naphthoquinone (5a) | 1,4...)
BDBM24776(1,4-Naphthoquinone | 1,4-Naphthoquinone (5a) | 1,4...)
BDBM24776(1,4-Naphthoquinone | 1,4-Naphthoquinone (5a) | 1,4...)
IC50: 8.40E+3nMAssay Description:The protocol for measuring IC50 values for the inhibition of MAO-A and MAO-B has been reported in detail in a recent publication (26). The recombinan...More data for this Ligand-Target Pair
BDBM24776(1,4-Naphthoquinone | 1,4-Naphthoquinone (5a) | 1,4...)
BDBM24776(1,4-Naphthoquinone | 1,4-Naphthoquinone (5a) | 1,4...)
BDBM24776(1,4-Naphthoquinone | 1,4-Naphthoquinone (5a) | 1,4...)
IC50: 1.10E+4nMAssay Description:Inhibition of recombinant AKT1 (unknown origin) using serine/threonine 06 peptide as substrate after 1 hr by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
BDBM24776(1,4-Naphthoquinone | 1,4-Naphthoquinone (5a) | 1,4...)
BDBM24776(1,4-Naphthoquinone | 1,4-Naphthoquinone (5a) | 1,4...)
IC50: 1.50E+4nMAssay Description:Inhibition of wild type human alpha-synuclein fibrillization expressed in Escherichia coli BL21(DE3)pLysS by thioflavin-T based fluorescence assayMore data for this Ligand-Target Pair
BDBM24776(1,4-Naphthoquinone | 1,4-Naphthoquinone (5a) | 1,4...)
BDBM24776(1,4-Naphthoquinone | 1,4-Naphthoquinone (5a) | 1,4...)
Papain(Carica papaya)Merck Research Laboratories
Curated by ChEMBL
BDBM24776(1,4-Naphthoquinone | 1,4-Naphthoquinone (5a) | 1,4...)
BDBM24776(1,4-Naphthoquinone | 1,4-Naphthoquinone (5a) | 1,4...)