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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
48
hits in this display
Target
Lysine-specific demethylase 4A
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
Ki: 4nM
Assay Description:
Binding affinity to KDM4A (unknown origin)
More data for this Ligand-Target Pair
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Target
Lysine-specific demethylase 4A
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
Ki: 4nM
Assay Description:
Binding affinity towards KDM4A (unknown origin)
More data for this Ligand-Target Pair
Target Info
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Target
Lysine-specific demethylase 5B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
Ki: 7nM
Assay Description:
Binding affinity to KDM5B (unknown origin)
More data for this Ligand-Target Pair
Target Info
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Target
Lysine-specific demethylase 5B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
Ki: 7nM
Assay Description:
Binding affinity towards KDM5B (unknown origin)
More data for this Ligand-Target Pair
Target Info
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Copy BDB DOI
Target
Lysine-specific demethylase 4B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5nM
Assay Description:
Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...
More data for this Ligand-Target Pair
Target Info
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Target
Lysine-specific demethylase 5B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5nM
Assay Description:
Inhibition of full length human KDM5B assessed as decrease in demethylation of substrate using peptide ARTK(me3)QTARKSTGGKAPRKQLA-GGK-biotin as subst...
More data for this Ligand-Target Pair
Target Info
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Copy BDB DOI
Target
Lysine-specific demethylase 5B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 7nM
Assay Description:
Inhibition of full length human KDM5B assessed as decrease in demethylation of substrate using peptide ARTK(me3)QTARKSTGGKAPRKQLA-GGK-biotin as subst...
More data for this Ligand-Target Pair
Target Info
PDB
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Copy BDB DOI
Target
Lysine-specific demethylase 4B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 8nM
Assay Description:
Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...
More data for this Ligand-Target Pair
Target Info
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Target
Lysine-specific demethylase 5B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 9nM
Assay Description:
Inhibition of full length human KDM5B assessed as decrease in demethylation of substrate using peptide ARTK(me3)QTARKSTGGKAPRKQLA-GGK-biotin as subst...
More data for this Ligand-Target Pair
Target Info
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Target
Lysine-specific demethylase 5B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 11nM
Assay Description:
Inhibition of full length human KDM5B assessed as decrease in demethylation of substrate using peptide ARTK(me3)QTARKSTGGKAPRKQLA-GGK-biotin as subst...
More data for this Ligand-Target Pair
Target Info
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Copy BDB DOI
Target
Lysine-specific demethylase 4B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 12nM
Assay Description:
Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...
More data for this Ligand-Target Pair
Target Info
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Copy BDB DOI
Target
Lysine-specific demethylase 4A
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 15nM
Assay Description:
Inhibition of full length human KDM4A A482E mutant assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbi...
More data for this Ligand-Target Pair
Target Info
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3D Structure (crystal)
Copy BDB DOI
Target
Lysine-specific demethylase 5B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 16nM
Assay Description:
Inhibition of full length human KDM5B assessed as decrease in demethylation of substrate using peptide ARTK(me3)QTARKSTGGKAPRKQLA-GGK-biotin as subst...
More data for this Ligand-Target Pair
Target Info
PDB
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Copy BDB DOI
Target
Lysine-specific demethylase 4A
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 22nM
Assay Description:
Inhibition of full length human KDM4A A482E mutant assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbi...
More data for this Ligand-Target Pair
Target Info
PDB
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UniProtKB/SwissProt
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Ligand Info
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In Depth
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PubMed
PDB
3D Structure (crystal)
Copy BDB DOI
Target
Lysine-specific demethylase 4B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 22nM
Assay Description:
Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...
More data for this Ligand-Target Pair
Target Info
PDB
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Copy BDB DOI
Target
Lysine-specific demethylase 5B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 23nM
Assay Description:
Inhibition of full length human KDM5B assessed as decrease in demethylation of substrate using peptide ARTK(me3)QTARKSTGGKAPRKQLA-GGK-biotin as subst...
More data for this Ligand-Target Pair
Target Info
PDB
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Copy BDB DOI
Target
Lysine-specific demethylase 4A
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 25nM
Assay Description:
Inhibition of full length human KDM4A A482E mutant assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbi...
More data for this Ligand-Target Pair
Target Info
PDB
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UniProtKB/SwissProt
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Ligand Info
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PDB
3D Structure (crystal)
Copy BDB DOI
Target
Lysine-specific demethylase 4B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 36nM
Assay Description:
Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...
More data for this Ligand-Target Pair
Target Info
PDB
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In Depth
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PubMed
Copy BDB DOI
Target
Lysine-specific demethylase 5B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 38nM
Assay Description:
Inhibition of KDM5B (unknown origin) assessed as decrease in demethylation of substrate using peptide (H3(1-21)K4-Me3-GGKBiotin) as substrate and 2OG...
More data for this Ligand-Target Pair
Target Info
PDB
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Copy BDB DOI
Target
Lysine-specific demethylase 5B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 39nM
Assay Description:
Inhibition of full length human KDM5B assessed as decrease in demethylation of substrate using peptide ARTK(me3)QTARKSTGGKAPRKQLA-GGK-biotin as subst...
More data for this Ligand-Target Pair
Target Info
PDB
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UniProtKB/SwissProt
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PC cid
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PDB
In Depth
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PubMed
Copy BDB DOI
Target
Lysine-specific demethylase 4A
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 39nM
Assay Description:
Inhibition of full length human KDM4A A482E mutant assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbi...
More data for this Ligand-Target Pair
Target Info
PDB
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UniProtKB/SwissProt
antibodypedia
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3D Structure (crystal)
Copy BDB DOI
Target
Lysine-specific demethylase 4B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 43nM
Assay Description:
Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...
More data for this Ligand-Target Pair
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Target
Lysine-specific demethylase 4A
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 61nM
Assay Description:
Inhibition of full length human KDM4A A482E mutant assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbi...
More data for this Ligand-Target Pair
Target Info
PDB
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3D Structure (crystal)
Copy BDB DOI
Target
Lysine-specific demethylase 4B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 62nM
Assay Description:
Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...
More data for this Ligand-Target Pair
Target Info
PDB
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Copy BDB DOI
Target
Lysine-specific demethylase 4B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 96nM
Assay Description:
Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...
More data for this Ligand-Target Pair
Target Info
PDB
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Copy BDB DOI
Target
Lysine-specific demethylase 4A
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 100nM
Assay Description:
Inhibition of N-terminal His-tagged recombinant human KDM4A (1 to 359 residues) expressed in Escherichia coli assessed as decrease in demethylation o...
More data for this Ligand-Target Pair
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Target
Lysine-specific demethylase 5B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 104nM
Assay Description:
Inhibition of full length human KDM5B assessed as decrease in demethylation of substrate using peptide ARTK(me3)QTARKSTGGKAPRKQLA-GGK-biotin as subst...
More data for this Ligand-Target Pair
Target Info
PDB
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Copy BDB DOI
Target
Lysine-specific demethylase 4A
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 114nM
Assay Description:
Inhibition of full length human KDM4A A482E mutant assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbi...
More data for this Ligand-Target Pair
Target Info
PDB
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Target
Lysine-specific demethylase 5C
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 123nM
Assay Description:
Inhibition of KDM5C (unknown origin) assessed as decrease in demethylation of substrate using peptide (H3(1-21)K4-Me3-GGKBiotin) as substrate and 2OG...
More data for this Ligand-Target Pair
Target Info
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MMDB
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KEGG
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Target
Lysine-specific demethylase 5B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 177nM
Assay Description:
Inhibition of full length human KDM5B assessed as decrease in demethylation of substrate using peptide ARTK(me3)QTARKSTGGKAPRKQLA-GGK-biotin as subst...
More data for this Ligand-Target Pair
Target Info
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Target
Lysine-specific demethylase 4A
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 197nM
Assay Description:
Inhibition of full length human KDM4A A482E mutant assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbi...
More data for this Ligand-Target Pair
Target Info
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Target
Lysine-specific demethylase 4B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 233nM
Assay Description:
Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...
More data for this Ligand-Target Pair
Target Info
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Target
Lysine-specific demethylase 5B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 371nM
Assay Description:
Inhibition of full length human KDM5B assessed as decrease in demethylation of substrate using peptide ARTK(me3)QTARKSTGGKAPRKQLA-GGK-biotin as subst...
More data for this Ligand-Target Pair
Target Info
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Target
Lysine-specific demethylase 4B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 382nM
Assay Description:
Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...
More data for this Ligand-Target Pair
Target Info
PDB
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Copy BDB DOI
Target
Lysine-specific demethylase 4A
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 423nM
Assay Description:
Inhibition of full length human KDM4A A482E mutant assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbi...
More data for this Ligand-Target Pair
Target Info
PDB
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3D Structure (crystal)
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Target
Lysine-specific demethylase 4B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
Copy InChI
Affinity Data
IC50: 524nM
Assay Description:
Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...
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Lysine-specific demethylase 4A
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
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Affinity Data
IC50: 657nM
Assay Description:
Inhibition of full length human KDM4A A482E mutant assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbi...
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Target
Lysine-specific demethylase 4B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
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Affinity Data
IC50: 787nM
Assay Description:
Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...
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Target
Lysine-specific demethylase 4A
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
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Affinity Data
IC50: 857nM
Assay Description:
Inhibition of full length human KDM4A A482E mutant assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbi...
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Target
Lysine-specific demethylase 5B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
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Affinity Data
IC50: 947nM
Assay Description:
Inhibition of full length human KDM5B assessed as decrease in demethylation of substrate using peptide ARTK(me3)QTARKSTGGKAPRKQLA-GGK-biotin as subst...
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Target
Lysine-specific demethylase 4A
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
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Affinity Data
IC50: 2.21E+3nM
Assay Description:
Inhibition of full length human KDM4A A482E mutant assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbi...
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Lysine-specific demethylase 2A
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
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IC50: 4.50E+3nM
Assay Description:
Inhibition of KDM2A (unknown origin) by Alphascreen assay
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Lysine-specific demethylase 3A
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
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IC50: 5.78E+3nM
Assay Description:
Inhibition of KDM3A (unknown origin) by Alphascreen assay
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Lysine-specific demethylase 6B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
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IC50: 9.02E+4nM
Assay Description:
Inhibition of KDM6B (unknown origin) by Alphascreen assay
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Lysine-specific demethylase 5B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
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Affinity Data
EC50: 1.34E+4nM
Assay Description:
Inhibition of full length human wild type KDM5B transfected in HeLa cells assessed as decrease in demethylation of H3K4Me3 measured after 24 hrs by c...
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Lysine-specific demethylase 5B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
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Affinity Data
EC50: 4.00E+3nM
Assay Description:
Binding affinity to recombinant human N-terminal KDM5B (26 to 772 residues) fused with ePL-tagged C-terminal transfected in HEK293T cells measured af...
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Lysine-specific demethylase 4B
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
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Affinity Data
EC50: 1.30E+3nM
Assay Description:
Binding affinity to recombinant human N-terminal KDM4B (1 to 348 residues) fused upstream with E31G-R71G-K105E/ePL-tagged C-terminal transfected in H...
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Target
Lysine-specific demethylase 4A
(Homo sapiens (Human))
Institute Of Cancer Research
Curated by
ChEMBL
Ligand
BDBM50513343
(CHEMBL4449500)
Copy SMILES
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Affinity Data
EC50: 4.70E+3nM
Assay Description:
Inhibition of FLAG tagged full length wild type human KDM4A transfected in HeLa cells assessed as decrease in demethylation of H3K9Me3 measured after...
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