Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 6 hits in this display
BDBM278181(2-(((3R,4S)-3-fluoro-1-((2S,4R)-4-hydroxy-5-oxopyr...)
BDBM278181(2-(((3R,4S)-3-fluoro-1-((2S,4R)-4-hydroxy-5-oxopyr...)
IC50: 6nMAssay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
BDBM278181(2-(((3R,4S)-3-fluoro-1-((2S,4R)-4-hydroxy-5-oxopyr...)
BDBM278181(2-(((3R,4S)-3-fluoro-1-((2S,4R)-4-hydroxy-5-oxopyr...)
BDBM278181(2-(((3R,4S)-3-fluoro-1-((2S,4R)-4-hydroxy-5-oxopyr...)
IC50: 6.00E+3nMpH: 7.0Assay Description:Enzymatic activity of IKKε and TBK1 was measured using a homogeneous time resolved fluorescence resonance energy transfer (TR-FRET) assay that m...More data for this Ligand-Target Pair
BDBM278181(2-(((3R,4S)-3-fluoro-1-((2S,4R)-4-hydroxy-5-oxopyr...)