Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 8 hits in this display
BDBM50444048(CHEMBL3092779 | US9649309, Compound UNC3053A)
BDBM50444048(CHEMBL3092779 | US9649309, Compound UNC3053A)
IC50: 82nMAssay Description:Briefly, activity assays were performed in a 384 well, polypropylene microplate in a final volume of 50 μL of 50 mM Hepes, Ph 7.4 containing 10 ...More data for this Ligand-Target Pair
BDBM50444048(CHEMBL3092779 | US9649309, Compound UNC3053A)
IC50: 83nMAssay Description:Inhibition of Mer kinase (unknown origin) using 5-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by microfluidic capillary electrophoresis assayMore data for this Ligand-Target Pair
BDBM50444048(CHEMBL3092779 | US9649309, Compound UNC3053A)
BDBM50444048(CHEMBL3092779 | US9649309, Compound UNC3053A)
IC50: 1.16E+3nMAssay Description:Briefly, activity assays were performed in a 384 well, polypropylene microplate in a final volume of 50 μL of 50 mM Hepes, Ph 7.4 containing 10 ...More data for this Ligand-Target Pair
BDBM50444048(CHEMBL3092779 | US9649309, Compound UNC3053A)
IC50: 1.32E+3nMAssay Description:Briefly, activity assays were performed in a 384 well, polypropylene microplate in a final volume of 50 μL of 50 mM Hepes, Ph 7.4 containing 10 ...More data for this Ligand-Target Pair
BDBM50444048(CHEMBL3092779 | US9649309, Compound UNC3053A)
IC50: 2.03E+4nMAssay Description:Briefly, activity assays were performed in a 384 well, polypropylene microplate in a final volume of 50 μL of 50 mM Hepes, Ph 7.4 containing 10 ...More data for this Ligand-Target Pair
BDBM50444048(CHEMBL3092779 | US9649309, Compound UNC3053A)
IC50: 2.03E+4nMAssay Description:Inhibition of Axl kinase (unknown origin) using 5-FAM-KKKKEEIYFFF-CONH2 as substrate after 180 mins by microfluidic capillary electrophoresis assayMore data for this Ligand-Target Pair