Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetD-alanyl-D-alanine carboxypeptidase(Actinomadura sp. (strain R39))
Universit£

Curated by ChEMBL
LigandPNGBDBM50385266(CHEMBL2035295)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of Actinomadura sp. R39 PBP using S2d as substrate incubated for 60 mins prior to substrate addition by DTNB-based spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPenicillin-binding protein 2X(Streptococcus pneumoniae R6)
Universit£

Curated by ChEMBL
LigandPNGBDBM50385266(CHEMBL2035295)
Affinity DataIC50:  4.81E+5nMAssay Description:Inhibition of penicillin-sensitive Streptococcus pneumoniae R6 PBP2x using S2d as substrate incubated for 60 mins prior to substrate addition by DTNB...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed