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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50314702((R)-2-(2-naphthamido)-5-(2-hydroxyphenyl)pent-4-yn...)
Affinity DataKi:  4.43E+3nMAssay Description:Displacement of WFYpSPFLE from human Pin1 catalytic domain after 10-20 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50314702((R)-2-(2-naphthamido)-5-(2-hydroxyphenyl)pent-4-yn...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human Pin1 by whole cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed