Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Free fatty acid receptor 2
(Homo sapiens (Human))
Epics Therapeutics
US Patent
Ligand
BDBM403842
((2S,5R)-5-(2-chlorophenyl)-1-(4-(pyridin-4-ylmetho...)
Copy SMILES
Copy InChI
Affinity Data
EC50: >1.00E+3nM
Assay Description:
The [35S]GTPγS assay was incubated in 20 mM HEPES pH7.4, 100 mM NaCl, 10 μg/ml saponin, 30 mM of MgCl2, 10 μM of GDP, 5 μg membra...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Free fatty acid receptor 2
(Homo sapiens (Human))
Epics Therapeutics
US Patent
Ligand
BDBM403842
((2S,5R)-5-(2-chlorophenyl)-1-(4-(pyridin-4-ylmetho...)
Copy SMILES
Copy InChI
Affinity Data
EC50: >1.00E+3nM
Assay Description:
The assay was used to determine the activity of the compounds of the invention. The [35S]GTPγS assay was incubated in 20 mM HEPES pH7.4, 100 mM ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Free fatty acid receptor 2
(Homo sapiens (Human))
Epics Therapeutics
US Patent
Ligand
BDBM403842
((2S,5R)-5-(2-chlorophenyl)-1-(4-(pyridin-4-ylmetho...)
Copy SMILES
Copy InChI
Affinity Data
EC50: >1.00E+3nM
Assay Description:
The assay was used to determine the activity of the compounds of the invention.The [35S]GTPγS assay was incubated in 20 mM HEPES pH7.4, 100 mM N...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Free fatty acid receptor 2
(Homo sapiens (Human))
Epics Therapeutics
US Patent
Ligand
BDBM403842
((2S,5R)-5-(2-chlorophenyl)-1-(4-(pyridin-4-ylmetho...)
Copy SMILES
Copy InChI
Affinity Data
EC50: >1.00E+3nM
Assay Description:
The following assay can be used for determination of GPR43 activation. When a GPCR is in its active state, either as a result of ligand binding or co...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI