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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
Lysophosphatidic acid receptor 2
(Homo sapiens (Human))
The University Of Memphis
Curated by
ChEMBL
Ligand
BDBM50271763
(3-[3-(3-Carboxy-acryloylamino)-phenylcarbamoyl]-ac...)
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Affinity Data
Ki: 20.8nM
Assay Description:
Antagonist activity at LPA2 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...
More data for this Ligand-Target Pair
Target Info
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Lysophosphatidic acid receptor 1
(Homo sapiens (Human))
The University Of Memphis
Curated by
ChEMBL
Ligand
BDBM50271763
(3-[3-(3-Carboxy-acryloylamino)-phenylcarbamoyl]-ac...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 50nM
Assay Description:
Antagonist activity at LPA1 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Lysophosphatidic acid receptor 2
(Homo sapiens (Human))
The University Of Memphis
Curated by
ChEMBL
Ligand
BDBM50271763
(3-[3-(3-Carboxy-acryloylamino)-phenylcarbamoyl]-ac...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 21.8nM
Assay Description:
Antagonist activity at LPA2 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...
More data for this Ligand-Target Pair
Target Info
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Lysophosphatidic acid receptor 2
(Homo sapiens (Human))
The University Of Memphis
Curated by
ChEMBL
Ligand
BDBM50271763
(3-[3-(3-Carboxy-acryloylamino)-phenylcarbamoyl]-ac...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 22nM
Assay Description:
Antagonist activity at LPA2 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium response
More data for this Ligand-Target Pair
Target Info
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Lysophosphatidic acid receptor 1
(Homo sapiens (Human))
The University Of Memphis
Curated by
ChEMBL
Ligand
BDBM50271763
(3-[3-(3-Carboxy-acryloylamino)-phenylcarbamoyl]-ac...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 220nM
Assay Description:
Antagonist activity at LPA1 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Lysophosphatidic acid receptor 1
(Homo sapiens (Human))
The University Of Memphis
Curated by
ChEMBL
Ligand
BDBM50271763
(3-[3-(3-Carboxy-acryloylamino)-phenylcarbamoyl]-ac...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 220nM
Assay Description:
Antagonist activity at LPA1 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium response
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI