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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetGlycogen phosphorylase, liver form(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50135552(4-{2-[(4-Chloro-pyridine-2-carbonyl)-amino]-phenox...)
Affinity DataIC50:  14nMAssay Description:Inhibitory activity against mouse liver glycogen phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50135552(4-{2-[(4-Chloro-pyridine-2-carbonyl)-amino]-phenox...)
Affinity DataIC50:  16nMAssay Description:Inhibitory activity against rat liver glycogen phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50135552(4-{2-[(4-Chloro-pyridine-2-carbonyl)-amino]-phenox...)
Affinity DataIC50:  17nMAssay Description:Inhibitory activity against HLGP(human liver glycogen phosphorylase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50135552(4-{2-[(4-Chloro-pyridine-2-carbonyl)-amino]-phenox...)
Affinity DataIC50:  181nMAssay Description:Inhibitory activity against HMGP(human muscle glycogen phosphorylase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed